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List of shared articles
Times cited
Discovery of N-Trisubstituted Pyrimidine Derivatives as Type I RET and RET Gatekeeper Mutant Inhibitors with a Novel Kinase Binding Pose.
Lingtian Zhang, Marialuisa Moccia, David C Briggs, Jaideep B Bharate, Naga Rajiv Lakkaniga, Phillip Knowles, Wei Yan, Phuc Tran, Anupreet Kharbanda, Xiuqi Wang,[...]. J Med Chem 2022
Lingtian Zhang, Marialuisa Moccia, David C Briggs, Jaideep B Bharate, Naga Rajiv Lakkaniga, Phillip Knowles, Wei Yan, Phuc Tran, Anupreet Kharbanda, Xiuqi Wang,[...]. J Med Chem 2022
Resistance to RET targeted therapy in Thyroid Cancer: Molecular basis and overcoming strategies.
María San Román-Gil, Javier Pozas, Diana Rosero-Rodríguez, Jesús Chamorro-Pérez, Álvaro Ruiz-Granados, Ignacio Ruz Caracuel, Enrique Grande, Javier Molina-Cerrillo, Teresa Alonso-Gordoa. Cancer Treat Rev 2022
María San Román-Gil, Javier Pozas, Diana Rosero-Rodríguez, Jesús Chamorro-Pérez, Álvaro Ruiz-Granados, Ignacio Ruz Caracuel, Enrique Grande, Javier Molina-Cerrillo, Teresa Alonso-Gordoa. Cancer Treat Rev 2022
The Emerging Portrait of Glial Cell Line-derived Neurotrophic Factor Family Receptor Alpha (GFRα) in Cancers.
Qingshang Li, Zhijun Cao, Shuliang Zhao. Int J Med Sci 2022
Qingshang Li, Zhijun Cao, Shuliang Zhao. Int J Med Sci 2022
ESMO recommendations on the standard methods to detect RET fusions and mutations in daily practice and clinical research.
C Belli, F Penault-Llorca, M Ladanyi, N Normanno, J-Y Scoazec, L Lacroix, J S Reis-Filho, V Subbiah, J F Gainor, V Endris,[...]. Ann Oncol 2021
C Belli, F Penault-Llorca, M Ladanyi, N Normanno, J-Y Scoazec, L Lacroix, J S Reis-Filho, V Subbiah, J F Gainor, V Endris,[...]. Ann Oncol 2021
Discovery and optimization of selective RET inhibitors via scaffold hopping.
Zhibo Luo, Lingli Wang, Zhifei Fu, Bin Shuai, Miaorong Luo, Guoping Hu, Jian Chen, Jikui Sun, Jiansong Wang, Jian Li,[...]. Bioorg Med Chem Lett 2021
Zhibo Luo, Lingli Wang, Zhifei Fu, Bin Shuai, Miaorong Luo, Guoping Hu, Jian Chen, Jikui Sun, Jiansong Wang, Jian Li,[...]. Bioorg Med Chem Lett 2021
Targeting Rearranged during Transfection in Cancer: A Perspective on Small-Molecule Inhibitors and Their Clinical Development.
Debasmita Saha, Katie Rose Ryan, Naga Rajiv Lakkaniga, Baku Acharya, Noemi Garcia Garcia, Erica Lane Smith, Brendan Frett. J Med Chem 2021
Debasmita Saha, Katie Rose Ryan, Naga Rajiv Lakkaniga, Baku Acharya, Noemi Garcia Garcia, Erica Lane Smith, Brendan Frett. J Med Chem 2021
Neuro-mesenchymal units control ILC2 and obesity via a brain-adipose circuit.
Filipa Cardoso, Roel G J Klein Wolterink, Cristina Godinho-Silva, Rita G Domingues, Hélder Ribeiro, Joaquim Alves da Silva, Inês Mahú, Ana I Domingos, Henrique Veiga-Fernandes. Nature 2021
Filipa Cardoso, Roel G J Klein Wolterink, Cristina Godinho-Silva, Rita G Domingues, Hélder Ribeiro, Joaquim Alves da Silva, Inês Mahú, Ana I Domingos, Henrique Veiga-Fernandes. Nature 2021
Hallmarks of RET and Co-occuring Genomic Alterations in RET-aberrant Cancers.
Jacob J Adashek, Aakash P Desai, Alexander Y Andreev-Drakhlin, Jason Roszik, Gilbert J Cote, Vivek Subbiah. Mol Cancer Ther 2021
Jacob J Adashek, Aakash P Desai, Alexander Y Andreev-Drakhlin, Jason Roszik, Gilbert J Cote, Vivek Subbiah. Mol Cancer Ther 2021
The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation.
Yuchen Jiang, Xia Peng, Yinchun Ji, Yang Dai, Yanfen Fang, Bing Xiong, Wenming Ren, Youhong Hu, Yi Chen, Jing Ai. Mol Cancer Ther 2021
Yuchen Jiang, Xia Peng, Yinchun Ji, Yang Dai, Yanfen Fang, Bing Xiong, Wenming Ren, Youhong Hu, Yi Chen, Jing Ai. Mol Cancer Ther 2021
[Advances in the Treatment of RET Fusion-positive Advanced Non-small Cell Lung Cancer].
Qingyun Gao, Junwei Su, Faman Xiao, Xiaocheng Lin, Jinji Yang. Zhongguo Fei Ai Za Zhi 2021
Qingyun Gao, Junwei Su, Faman Xiao, Xiaocheng Lin, Jinji Yang. Zhongguo Fei Ai Za Zhi 2021
PTPRA Phosphatase Regulates GDNF-Dependent RET Signaling and Inhibits the RET Mutant MEN2A Oncogenic Potential.
Leena Yadav, Elina Pietilä, Tiina Öhman, Xiaonan Liu, Arun K Mahato, Yulia Sidorova, Kaisa Lehti, Mart Saarma, Markku Varjosalo. iScience 2020
Leena Yadav, Elina Pietilä, Tiina Öhman, Xiaonan Liu, Arun K Mahato, Yulia Sidorova, Kaisa Lehti, Mart Saarma, Markku Varjosalo. iScience 2020
Targeting RET Kinase in Neuroendocrine Prostate Cancer.
Halena R VanDeusen, Johnny R Ramroop, Katherine L Morel, Song Yi Bae, Anjali V Sheahan, Zoi Sychev, Nathan A Lau, Larry C Cheng, Victor M Tan, Zhen Li,[...]. Mol Cancer Res 2020
Halena R VanDeusen, Johnny R Ramroop, Katherine L Morel, Song Yi Bae, Anjali V Sheahan, Zoi Sychev, Nathan A Lau, Larry C Cheng, Victor M Tan, Zhen Li,[...]. Mol Cancer Res 2020
Progresses Toward Precision Medicine in RET-altered Solid Tumors.
Carmen Belli, Santosh Anand, Justin F Gainor, Frederique Penault-Llorca, Vivek Subbiah, Alexander Drilon, Fabrice Andrè, Giuseppe Curigliano. Clin Cancer Res 2020
Carmen Belli, Santosh Anand, Justin F Gainor, Frederique Penault-Llorca, Vivek Subbiah, Alexander Drilon, Fabrice Andrè, Giuseppe Curigliano. Clin Cancer Res 2020
Discovery of 4-methyl-N-(4-((4-methylpiperazin- 1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-oxy)benzamide as a potent inhibitor of RET and its gatekeeper mutant.
Xiaoyang Li, Jingyi Su, Yanru Yang, Wenhua Lian, Zhou Deng, Zaiyou Yang, Guyue Chen, Baoding Zhang, Chao Dong, Xueyan Liu,[...]. Eur J Med Chem 2020
Xiaoyang Li, Jingyi Su, Yanru Yang, Wenhua Lian, Zhou Deng, Zaiyou Yang, Guyue Chen, Baoding Zhang, Chao Dong, Xueyan Liu,[...]. Eur J Med Chem 2020
Targeted therapies for RET-fusion cancer: Dilemmas and breakthrough.
SiJie Ding, Rong Wang, ShunLi Peng, Xiaoqing Luo, LongHui Zhong, Hong Yang, YueYun Ma, ShiYu Chen, Wei Wang. Biomed Pharmacother 2020
SiJie Ding, Rong Wang, ShunLi Peng, Xiaoqing Luo, LongHui Zhong, Hong Yang, YueYun Ma, ShiYu Chen, Wei Wang. Biomed Pharmacother 2020