K M Kim, S F Kingsmore, H Han, T L Yang-Feng, N Godinot, M F Seldin, M G Caron, B Giros. Mol Pharmacol 1994
Times Cited: 154
Times Cited: 154
B N Atkinson, S C Bell, M De Vivo, L R Kowalski, S M Lechner, V I Ognyanov, C S Tham, C Tsai, J Jia, D Ashton, M A Klitenick. Mol Pharmacol 2001
Times Cited: 148
Times Cited: 148
List of shared articles
Times cited
Reduction of Rapid Proliferating Tumour Cell Lines by Inhibition of the Specific Glycine Transporter GLYT1.
Christine Garcia Bierhals, Alison Howard, Barry H Hirst. Biomedicines 2021
Christine Garcia Bierhals, Alison Howard, Barry H Hirst. Biomedicines 2021
A System for Assessing Dual Action Modulators of Glycine Transporters and Glycine Receptors.
Diba Sheipouri, Casey I Gallagher, Susan Shimmon, Tristan Rawling, Robert J Vandenberg. Biomolecules 2020
Diba Sheipouri, Casey I Gallagher, Susan Shimmon, Tristan Rawling, Robert J Vandenberg. Biomolecules 2020
Time-dependent impact of glutamatergic modulators on the promnesiant effect of 5-HT6R blockade on mice recognition memory.
Rachel Asselot, Emmanuelle Simon-O'Brien, Sophie Lebourgeois, Gérald Nee, Virgile Delaunay, Pascal Duchatelle, Valentine Bouet, François Dauphin. Pharmacol Res 2017
Rachel Asselot, Emmanuelle Simon-O'Brien, Sophie Lebourgeois, Gérald Nee, Virgile Delaunay, Pascal Duchatelle, Valentine Bouet, François Dauphin. Pharmacol Res 2017
Inhibitors of Glycine Transporter-1: Potential Therapeutics for the Treatment of CNS Disorders.
Christopher L Cioffi, Peter R Guzzo. Curr Top Med Chem 2016
Christopher L Cioffi, Peter R Guzzo. Curr Top Med Chem 2016
Lipid inhibitors of high affinity glycine transporters: identification of a novel class of analgesics.
Jane E Carland, Cheryl A Handford, Renae M Ryan, Robert J Vandenberg. Neurochem Int 2014
Jane E Carland, Cheryl A Handford, Renae M Ryan, Robert J Vandenberg. Neurochem Int 2014
Oleoyl-L-carnitine inhibits glycine transport by GlyT2.
J E Carland, R E Mansfield, R M Ryan, R J Vandenberg. Br J Pharmacol 2013
J E Carland, R E Mansfield, R M Ryan, R J Vandenberg. Br J Pharmacol 2013
Amino-terminal isoforms of the human glycine transporter GlyT1 exhibit similar pharmacology.
John T Durkin, Chrysanthe M Spais, Justin Schreiber, Karla Kopec, Sheryl L Meyer. Brain Res 2011
John T Durkin, Chrysanthe M Spais, Justin Schreiber, Karla Kopec, Sheryl L Meyer. Brain Res 2011
In vivo evaluation of carbon-11-labelled non-sarcosine-based glycine transporter 1 inhibitors in mice and conscious monkeys.
Jun Toyohara, Kiichi Ishiwata, Muneyuki Sakata, Jin Wu, Shingo Nishiyama, Hideo Tsukada, Kenji Hashimoto. Nucl Med Biol 2011
Jun Toyohara, Kiichi Ishiwata, Muneyuki Sakata, Jin Wu, Shingo Nishiyama, Hideo Tsukada, Kenji Hashimoto. Nucl Med Biol 2011
The glycine transporter GLYT1 in human intestine: expression and function.
Alison Howard, Barry Hugo Hirst. Biol Pharm Bull 2011
Alison Howard, Barry Hugo Hirst. Biol Pharm Bull 2011
SLC6 neurotransmitter transporters: structure, function, and regulation.
Anders S Kristensen, Jacob Andersen, Trine N Jørgensen, Lena Sørensen, Jacob Eriksen, Claus J Loland, Kristian Strømgaard, Ulrik Gether. Pharmacol Rev 2011
Anders S Kristensen, Jacob Andersen, Trine N Jørgensen, Lena Sørensen, Jacob Eriksen, Claus J Loland, Kristian Strømgaard, Ulrik Gether. Pharmacol Rev 2011
Recent progress in the discovery of non-sarcosine based GlyT1 inhibitors.
Scott E Wolkenberg, Cyrille Sur. Curr Top Med Chem 2010
Scott E Wolkenberg, Cyrille Sur. Curr Top Med Chem 2010
Glycine transport inhibitors for the treatment of schizophrenia.
Kenji Hashimoto. Open Med Chem J 2010
Kenji Hashimoto. Open Med Chem J 2010
Glycine transporter inhibitors as a novel drug discovery strategy for neuropathic pain.
Toshihiro Dohi, Katsuya Morita, Tomoya Kitayama, Naoyo Motoyama, Norimitsu Morioka. Pharmacol Ther 2009
Toshihiro Dohi, Katsuya Morita, Tomoya Kitayama, Naoyo Motoyama, Norimitsu Morioka. Pharmacol Ther 2009
The phosphatidylinositol 3-kinase inhibitor LY 294002 inhibits GlyT1-mediated glycine uptake.
Zhi-Liang Wu, Teresa M O'Kane, Thomas J Connors, Michael J Marino, Hervé Schaffhauser. Brain Res 2008
Zhi-Liang Wu, Teresa M O'Kane, Thomas J Connors, Michael J Marino, Hervé Schaffhauser. Brain Res 2008
Inhibitors of GlyT1 affect glycine transport via discrete binding sites.
Mario Mezler, Wilfried Hornberger, Reinhold Mueller, Martin Schmidt, Willi Amberg, Wilfried Braje, Michael Ochse, Hans Schoemaker, Berthold Behl. Mol Pharmacol 2008
Mario Mezler, Wilfried Hornberger, Reinhold Mueller, Martin Schmidt, Willi Amberg, Wilfried Braje, Michael Ochse, Hans Schoemaker, Berthold Behl. Mol Pharmacol 2008
Design of potent GlyT1 inhibitors: in vitro and in vivo profiles.
Thomas M Bridges, Richard Williams, Craig W Lindsley. Curr Opin Mol Ther 2008
Thomas M Bridges, Richard Williams, Craig W Lindsley. Curr Opin Mol Ther 2008
Molecular basis for substrate discrimination by glycine transporters.
Robert J Vandenberg, Kim Shaddick, Pengchu Ju. J Biol Chem 2007
Robert J Vandenberg, Kim Shaddick, Pengchu Ju. J Biol Chem 2007
Glycine transporter 1 inhibitors and modulation of NMDA receptor-mediated excitatory neurotransmission.
Cyrille Sur, Gene G Kinney. Curr Drug Targets 2007
Cyrille Sur, Gene G Kinney. Curr Drug Targets 2007
Glutamate-based therapeutic approaches: inhibitors of glycine transport.
Sandra M Lechner. Curr Opin Pharmacol 2006
Sandra M Lechner. Curr Opin Pharmacol 2006
Development of a novel high-throughput assay for the investigation of GlyT-1b neurotransmitter transporter function.
Lynda Allan, J Lianne Leith, Marianthi Papakosta, John A Morrow, Nicholas G Irving, Brian W McFerran, Alan G Clark. Comb Chem High Throughput Screen 2006
Lynda Allan, J Lianne Leith, Marianthi Papakosta, John A Morrow, Nicholas G Irving, Brian W McFerran, Alan G Clark. Comb Chem High Throughput Screen 2006
Glycine transporter type-1 and its inhibitors.
L G Harsing, Z Juranyi, I Gacsalyi, P Tapolcsanyi, A Czompa, P Matyus. Curr Med Chem 2006
L G Harsing, Z Juranyi, I Gacsalyi, P Tapolcsanyi, A Czompa, P Matyus. Curr Med Chem 2006
Pharmacological properties of glycine uptake in the developing rat retina.
Rocío Salceda. Neurochem Int 2006
Rocío Salceda. Neurochem Int 2006
Progress towards validating the NMDA receptor hypofunction hypothesis of schizophrenia.
Craig W Lindsley, William D Shipe, Scott E Wolkenberg, Cory R Theberge, David L Williams, Cyrille Sur, Gene G Kinney. Curr Top Med Chem 2006
Craig W Lindsley, William D Shipe, Scott E Wolkenberg, Cory R Theberge, David L Williams, Cyrille Sur, Gene G Kinney. Curr Top Med Chem 2006
Design, synthesis, and in vivo efficacy of glycine transporter-1 (GlyT1) inhibitors derived from a series of [4-phenyl-1-(propylsulfonyl)piperidin-4-yl]methyl benzamides.
Craig W Lindsley, Zhijian Zhao, William H Leister, Julie O'Brien, Wei Lemaire, David L Williams, Tsing-Bau Chen, Raymond S L Chang, Maryann Burno, Marlene A Jacobson,[...]. ChemMedChem 2006
Craig W Lindsley, Zhijian Zhao, William H Leister, Julie O'Brien, Wei Lemaire, David L Williams, Tsing-Bau Chen, Raymond S L Chang, Maryann Burno, Marlene A Jacobson,[...]. ChemMedChem 2006
Progress in the preparation and testing of glycine transporter type-1 (GlyT1) inhibitors.
Craig W Lindsley, Scott E Wolkenberg, Gene G Kinney. Curr Top Med Chem 2006
Craig W Lindsley, Scott E Wolkenberg, Gene G Kinney. Curr Top Med Chem 2006
Neurochemical, electrophysiological and pharmacological profiles of the selective inhibitor of the glycine transporter-1 SSR504734, a potential new type of antipsychotic.
Ronan Depoortère, Gihad Dargazanli, Genevieve Estenne-Bouhtou, Annick Coste, Christophe Lanneau, Christophe Desvignes, Martine Poncelet, Michel Heaulme, Vincent Santucci, Michel Decobert,[...]. Neuropsychopharmacology 2005
Ronan Depoortère, Gihad Dargazanli, Genevieve Estenne-Bouhtou, Annick Coste, Christophe Lanneau, Christophe Desvignes, Martine Poncelet, Michel Heaulme, Vincent Santucci, Michel Decobert,[...]. Neuropsychopharmacology 2005
The therapeutic potential of glycine transporter-1 inhibitors.
Cyrille Sur, Gene G Kinney. Expert Opin Investig Drugs 2004
Cyrille Sur, Gene G Kinney. Expert Opin Investig Drugs 2004
Allosteric modulation of neurotransmitter transporters at excitatory synapses.
Robert J Vandenberg, Pengchu Ju, Karin R Aubrey, Renae M Ryan, Ann D Mitrovic. Eur J Pharm Sci 2004
Robert J Vandenberg, Pengchu Ju, Karin R Aubrey, Renae M Ryan, Ann D Mitrovic. Eur J Pharm Sci 2004
Arachidonic acid and anandamide have opposite modulatory actions at the glycine transporter, GLYT1a.
Rhonda Jo Pearlman, Karin R Aubrey, Robert J Vandenberg. J Neurochem 2003
Rhonda Jo Pearlman, Karin R Aubrey, Robert J Vandenberg. J Neurochem 2003
Glycine tranporter-1 blockade potentiates NMDA-mediated responses in rat prefrontal cortical neurons in vitro and in vivo.
Long Chen, Mark Muhlhauser, Charles R Yang. J Neurophysiol 2003
Long Chen, Mark Muhlhauser, Charles R Yang. J Neurophysiol 2003
Pharmacology and expression analysis of glycine transporter GlyT1 with [3H]-(N-[3-(4'-fluorophenyl)-3-(4'phenylphenoxy)propyl])sarcosine.
Pierre J Mallorga, Jacinta B Williams, Marlene Jacobson, Rosemary Marques, Ashok Chaudhary, P Jeffrey Conn, Douglas J Pettibone, Cyrille Sur. Neuropharmacology 2003
Pierre J Mallorga, Jacinta B Williams, Marlene Jacobson, Rosemary Marques, Ashok Chaudhary, P Jeffrey Conn, Douglas J Pettibone, Cyrille Sur. Neuropharmacology 2003
Development of a scintillation proximity assay for analysis of Na+/Cl- -dependent neurotransmitter transporter activity.
Jacinta B Williams, Pierre J Mallorga, Wei Lemaire, David L Williams, Sang Na, Smita Patel, P Jeffrey Conn, Douglas J Pettibone, Christopher Austin, Cyrille Sur. Anal Biochem 2003
Jacinta B Williams, Pierre J Mallorga, Wei Lemaire, David L Williams, Sang Na, Smita Patel, P Jeffrey Conn, Douglas J Pettibone, Christopher Austin, Cyrille Sur. Anal Biochem 2003
Glycine transporter isoforms in the mammalian central nervous system: structures, functions and therapeutic promises.
Jesus Gomeza, Koji Ohno, Heinrich Betz. Curr Opin Drug Discov Devel 2003
Jesus Gomeza, Koji Ohno, Heinrich Betz. Curr Opin Drug Discov Devel 2003
Structure, function and regulation of glycine neurotransporters.
Carmen Aragón, Beatriz López-Corcuera. Eur J Pharmacol 2003
Carmen Aragón, Beatriz López-Corcuera. Eur J Pharmacol 2003
Why glycine transporters have different stoichiometries.
Stéphane Supplisson, Michel J Roux. FEBS Lett 2002
Stéphane Supplisson, Michel J Roux. FEBS Lett 2002